SB269970 HCl

CAS No. 261901-57-9

SB269970 HCl ( SB-269970A )

Catalog No. M17459 CAS No. 261901-57-9

SB269970 HCl, a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity against other receptors.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 45 In Stock
5MG 61 In Stock
10MG 113 In Stock
25MG 243 In Stock
50MG 426 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    SB269970 HCl
  • Note
    Research use only, not for human use.
  • Brief Description
    SB269970 HCl, a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity against other receptors.
  • Description
    SB269970 HCl, a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity against other receptors.
  • Synonyms
    SB-269970A
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    5-HT7
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    261901-57-9
  • Formula Weight
    388.95
  • Molecular Formula
    C18H28N2O3S·HCl
  • Purity
    98%
  • Solubility
    DMSO : ≥ 30 mg/mL; 77.13 mM
  • SMILES
    Cl.CC1CCN(CC[C@H]2CCCN2S(=O)(=O)c2cccc(O)c2)CC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Hagan JJ, et al. Br J Pharmacol, 2000, 130(3), 539-548.
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