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SB269970 HCl

CAS No. 261901-57-9

SB269970 HCl ( SB-269970A )

Catalog No. M17459 CAS No. 261901-57-9

SB269970 HCl, a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity against other receptors.

Purity : 98%

COA

Datasheet

HNMR

HPLC

MSDS

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Size	Price / USD	Stock	Quantity
2MG	45	In Stock
5MG	61	In Stock
10MG	113	In Stock
25MG	243	In Stock
50MG	426	In Stock
100MG	Get Quote	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

SB269970 HCl
Note

Research use only, not for human use.
Brief Description

SB269970 HCl, a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity against other receptors.
Description

SB269970 HCl, a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity against other receptors.
Synonyms

SB-269970A
Pathway

Membrane Transporter/Ion Channel
Target

TRP/TRPV Channel
Recptor

5-HT7
Research Area

Neurological Disease
Indication

——

Chemical Information

CAS Number

261901-57-9
Formula Weight

388.95
Molecular Formula

C18H28N2O3S·HCl
Purity

98%
Solubility

DMSO : ≥ 30 mg/mL; 77.13 mM
SMILES

Cl.CC1CCN(CC[C@H]2CCCN2S(=O)(=O)c2cccc(O)c2)CC1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Hagan JJ, et al. Br J Pharmacol, 2000, 130(3), 539-548.

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